货号 | CAS号 |
---|---|
O127787-100mg | 686344-29-6 |
O127787-25mg | 686344-29-6 |
O127787-5mg | 686344-29-6 |
溶解性 | DMSO |
存贮条件 | 储存温度-20°C |
产品介绍 | Otenabant (CP945598)是CB1受体高亲和性拮抗剂,Ki为0.7 nM。 |
生化机理 | Otenabant (CP-945,598) exhibits sub-nanomolar potency at human CB1 receptors in both binding (Ki = 0.7 nM) and functional assays (Ki = 0.2 nM). The compound has low affinity (Ki = 7600 nM) for human CB2 receptors. |
别名 | 奥替那班; 1-[9-(4-氯苯基)-8-(2-氯苯基)-9H-嘌呤-6-基]-4-乙基氨基哌啶-4-甲酰胺;CP 945598;CP-945598;CP945598;1-[9-(4-Chlorophenyl)-8-(2-chlorophenyl)-9H-purin-6-yl]-4-ethylaminopiperidine-4-carboxamide |