AG-879

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AG-879, a member of the tyrphostin family of tyrosine kinase inhibitors, inhibits NGF receptor (pp140c-trk) autophosphorylation selectively with no inhibition of EGF or PDGF receptor phosphorylation (IC50=10 µM). AG-879 inhibits NGF-induced neurite outgrowth in PC12 cells.
Product Specification
Formula: C18H24N2OS
MW: 316.5
Purity: ≥99%
Appearance: Yellow solid.
CAS: 148741-30-4
Solubility: Soluble in 100% ethanol (25mg/ml) or DMSO (25mg/ml).
Shipping: AMBIENT
Long Term Storage: -20°C
Handling: Protect from light.
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