溶解性 |
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存贮条件 | 储存温度-20°C |
产品介绍 | TAE226 (NVP-TAE226)是一种有效的FAK抑制剂,IC50为5.5 nM,最有效作用于Pyk2,对InsR, IGF-1R, ALK和c-Met作用效果比其弱10到100倍左右 |
备注 | NVP-TAE226 is a potent FAK inhibitor with IC50 of 5.5 nM and modestly potent to Pyk2, ~10- to 100-fold less potent against InsR, IGF-1R, ALK, and c-Met. |
生化机理 |
NVP-TAE 226(TAE226) is a potent dual FAK/IGF-IR kinase inhibitor. |
别名 | 2-[[5-氯-2-[[2-甲氧基-4-(4-吗啉基)苯基]氨基]-4-嘧啶基]氨基]-N-甲基苯甲酰胺;2-[[5-Chloro-2-[[2-methoxy-4-(4-morpholinyl)phenyl]amino]-4-pyrimidinyl]amino]-N-methylbenzamide |