敏感性 | 对热、光线敏感 |
溶解性 |
, |
存贮条件 | 储存温度-20°C |
应用 | A selective SR-1B/SR-1D |
产品介绍 | Eletriptan HBr 是一种选择性的5-羟色胺1B和1D受体激动剂,Ki值分别为0.92 nM和3.14 nM。 |
备注 | Eletriptan is a selective 5-HT1B and 5-HT1D receptor agonist with Ki of 0.92 nM and 3.14 nM, respectively. |
生化机理 | Eletriptan hydrobromide is a selective SR-1B/SR-1D agonist. |
别名 | N/A;依来曲普坦氢溴酸盐; 来曲普坦氢溴酸盐; 依利曲坦氢溴酸盐; (R)-3-[(1-甲基-2-吡咯烷基)甲基]-5-[2-(苯磺酰)乙基]-1H-吲哚氢溴酸盐;N/A;Eletriptan hydrobromide;3-(((2R)-1-Methyl-2-pyrrolidinyl))methyl)-5-(2-(phenylsulfonyl)ethyl)-1H-indole hydrobromide |