熔点 | 160 °C |
溶解性 | Soluble in water, methanol, and DMSO. |
存贮条件 | 储存温度 2-8°C |
应用 | An α2-adrenergic agonist. |
产品介绍 | Detomidine HCl可产生镇静和镇痛作用,这种作用具有剂量依赖性,通过激活α2儿茶酚胺受体来调节。 |
备注 | Detomidine produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors. |
生化机理 | Detomidine HCl is a nonnarcotic, synthetic alpha-2 adrenoreceptor agonist. Alpha2-adrenergic agonists produce dose-dependent sedative and analgesic effects, mediatated by activation of alpha-2 catecholamine receptors, thus inducing a negative feedback response, reducing production of excitatory neurotransmitters. |
别名 | 地托咪定盐酸盐;5-(2,3-二甲苯基)-1H-咪唑盐酸盐;盐酸地托咪定; 4-[(2,3-二甲基苯基)甲基]-1H-咪唑盐酸盐;5-(2,3-Dimethylbenzyl)-1H-imidazole Hydrochloride;Detomidine Hydrochloride;4-[(2,3-Dimethylphenyl)methyl]-1H-imidazole monohydrochloride;Detomidine hydrochloride |