溶解性 | Soluble in ethanol (77 mg/ml at 25 °C), DMSO (≥44 mg/ml), and water (<1 mg/ml at 25 °C). |
应用 | A potent enkephalinase inhibitor which exhibits selective antisecretory activity. |
产品介绍 | Racecadotril 是一种外周性的脑啡肽酶抑制剂,IC50为4.5 μM。 |
备注 | Racecadotril is a peripherally acting enkephalinase inhibitor with an IC50 of 4.5 μM |
生化机理 | Racecadotril is a potent CD10 (enkephalinase) inhibitor which exhibits selective antisecretory activity. |
别名 | 消旋卡多曲;醋托泛;N-[3-(乙酰基硫代)-2-苯丙酰基]甘氨酸苯甲酯;Acetorphan;Benzyl N-[3-(Acetylthio)-2-benzylpropionyl]glycinate;N-[3-(Acetylthio)-2-benzylpropionyl]glycine Benzyl Ester;(±)-Acetorphan;(RS)-Benzyl N-[3-(acetylthio)-2-benzylpropanoyl]glycinate;Cadotril;Redotil;Tiorfan;Zedott |