溶解性 | Soluble in DMSO (100 mM), and ethanol (10 mM). |
存贮条件 | 储存温度 2-8°C |
应用 | A selective SR-4 activator and a SR-3 inhibitor. |
产品介绍 | Mosapride Citrate是一种促胃肠动力药,是选择性5HT4激动剂。 |
备注 | Mosapride Citrate is a gastroprokinetic agent that acts as a selective 5HT4 agonist. |
生化机理 | Mosapride citrate is a selective SR-4 agonist and SR-3 antagonist. Increases gastric emptying in rats and stimulates gastric motor activity in conscious dogs. |
别名 | 枸橼酸莫沙必利; 4-氨基-5-氯-2-乙氧基-N-[[4-(4-氟苄基)-2-吗啉基]甲基]苯甲酰胺枸橼酸盐;Moza citrate; TAK-370 citrate; AS-4370 citrate; Gasmotin citrate;4-Amino-5-chloro-2-ethoxy-N-[[4-[(4-fluorophenyl)methyl]-2-morpholinyl]methyl]-benzamide 2-hydroxy-1,2,3-propanetricarboxylate |