溶解性 | DMSO ≥80mg/mL Water <1.2mg/mL Ethanol <1.2mg/mL |
存贮条件 | 储存温度-20°C |
应用 | An inhibitor of JAK1 and JAK2. |
产品介绍 | Momelotinib (CYT387)是一种ATP竞争性JAK1/JAK2抑制剂,IC50为11 nM/18 nM,比作用于JAK3选择性约高10倍左右。 |
生化机理 | Cyt387 is an ATP competitive inhibitor of JAK1 (IC50 = 11 nM) and JAK2 (IC50 = 18 nM) (Janus kinases). |
别名 | CYT 387; CYT-387;N-(氰基甲基)-4-[2-[[4-(4-吗啉基)苯基]氨基]-4-嘧啶基]苯甲酰胺;CYT 387; CYT-387;Momelotinib;N-(Cyanomethyl)-4-[2-[[4-(4-morpholinyl)phenyl]amino]-4-pyrimidinyl]benzamide |