敏感性 | 对光敏感 |
溶解性 | DMSO : 6.25 mg/mL |
存贮条件 | 储存温度-20°C |
密度 | 1.2800 |
应用 | 钙调蛋白(Ca2+-calmodulin)依赖的磷酸二酯酶I(PDE1)抑制剂。 |
产品介绍 | 不溶于水,溶于DMSO. |
生化机理 |
Vinpocetine(Cavinton; Ethyl apovincaminate;) is a phosphodiesterase inhibitor. Vinpocetine(Cavinton; Ethyl apovincaminate;) is selective for PDE1 (IC50 = 21 μM). Also blocks voltage-gated Na+ channels. |
别名 | 长春西汀 ;阿扑长春胺酸乙酯;Eburnamenine-14-carboxylic acid ethyl ester (3α, 16α)-Eburnamenine-14-carboxylic acid ethyl ester |