产品描述
| 熔点 | 157°C |
| 溶解性 | DMSO: ~14 mg/mL；H2O: insoluble |
| 应用 | Tofisopam has been used for studying its biochemical mechanisms of actions using drug repositioning strategies1. |
| 生化机理 | Ligand for the GABAA receptor benzodiazepine modulatory site. Studies have reported that tofisopam functions by blocking PDE4 (phosphodiesterase 4). Furthermore, the S-enantiomer of tofisopam is considered ten times more active than R-enantiomer |
| 别名 | 托非索泮; 1-(3,4-二甲氧基苯基)-5-乙基-7,8-二甲氧基-4-甲基-5H-苯并[d][1,2]二氮杂卓; 1-(3,4-二甲氧基苯基)-5-乙基-7,8-二甲氧基-4-甲基-5H-2,3-苯并二氮杂卓;1-(3,4-Dimethoxyphenyl)-5-ethyl-7,8-dimethoxy-4-methyl-5H-benzo[d][1,2]diazepine; 1-(3,4-Dimethoxyphenyl)-5-ethyl-7,8-dimethoxy-4-methyl-5H-2,3-benzodiazepine; Tofisopam；7,8-Dimethoxy-1-(3,4-dimethoxyphenyl)-5-ethyl-4-methyl-5H-2,3-benzodiazepine； EGYT 341； Seriel |
