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CAS No. : 1872466-47-1
MCE 国际站:CM-675
产品活性:CM-675 是磷酸二酯酶 5 (PDE5)和I类组蛋白去乙酰化酶 (HDAC1) 的选择性抑制剂,其对 PDE5 和 HDAC1 的IC50 值分别为114 nM 和673 nM。CM-675 可用于阿尔兹海默症的研究。
研究领域:Metabolic Enzyme/Protease | Epigenetics | Cell Cycle/DNA Damage
作用靶点:Phosphodiesterase (PDE) | HDAC
In Vitro: CM-675 (29a) shows a significant time-dependent effect on class I HDAC inhibition, particularly towards HDAC2. For HDAC1, its inhibitory potency also increased significantly (~1 log unit) with the pre-incubation time: 673 nM (30 min), 180 nM (4 hours) and 69 nM (6 hours) .
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