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CAS No. : 1714146-59-4
MCE 国际站:I-BRD9
产品活性:I-BRD9 是含溴结构域蛋白 9 (BRD9) 的选择性细胞化学探针,其 pIC50 值为 7.3 μM。I-BRD9 对溴结构域和额外末端结构域 (BET) 家族和高度同源的含溴结构域蛋白 7 (BRD7) 具有很高的选择性。I-BRD9 可用于识别Kasumi-1 细胞中受 BRD9 调控的参与肿瘤和免疫应答通路的基因。
研究领域:Epigenetics
In Vitro: I-BRD9 (10 μM, 6 h) has a regulation role in cancer and immunology pathways.
I-BRD9 (10 μM) has high BRD9 affinity and excellent broader bromodomain selectivity.
I-BRD9 (10 μM) has affinity for BRD9 (TR-FRET), BRD4 BD1 (TR-FRET) and BRD9 NanoBRET with pIC50 values of 7.3 μM, 5.3 μM and 6.8 μM.
I-BRD9 (10 μM) has high aqueous solubility (CLND) with 359 μM.
I-BRD9 (10 μM) displays >625 fold selectivity in binding with endogenous BRD9 against BET family member BRD3 in HUT-78 cell lysate.
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