货号 | CAS号 |
---|---|
M126898-10mg | 606143-89-9 |
M126898-50mg | 606143-89-9 |
溶解性 |
|
存贮条件 | 储存温度-20°C |
备注 | ARRY-438162 is a potent inhibitor of MEK1/2 with IC50 of 12 nM. |
生化机理 |
MEK162(ARRY-162; ARRY-438162) is an oral, highly selective MEK inhibitor. MEK162(ARRY-162; ARRY-438162) is now being investigated in Phase I trials in advanced solid tumors. |
别名 | 1H-Benzimidazole-6-carboxamide, 5-[(4-bromo-2-fluorophenyl)amino]-4-fluoro-N-(2-hydroxyethoxy)-1-methyl-;1H-Benzimidazole-6-carboxamide, 5-[(4-bromo-2-fluorophenyl)amino]-4-fluoro-N-(2-hydroxyethoxy)-1-methyl- |