| 货号 | CAS号 |
|---|---|
| G129554-10mg | 309712-55-8 |
| G129554-50mg | 309712-55-8 |
| 溶解性 |
|
| 存贮条件 | 储存温度-20°C |
| 备注 | GW791343 HCl is aHCl salt form of GW791343, which is a non-competitive allosteric modulator of human P2X7 receptor inhibitor with pIC50 of 7. |
| 生化机理 |
GW791343 is a P2X7 allosteric modulator. Exhibits species-specific activity and acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2). A positive allosteric modulator of rat P2X7. |
| 别名 | 2-[(3,4-二氟苯基)氨基]-N-[2-甲基-5-(1-哌嗪基甲基)苯基]乙酰胺盐酸盐 ;2-[(3,4-Difluorophenyl)amino]-N-[2-methyl-5-(1-piperazinylmethyl)phenyl]acetamide hydrochloride |
