| 应用 |
A histamine H1 receptors antagonist |
| 产品介绍 |
Brompheniramine hydrogen maleate是一种组胺H1受体拮抗剂。 |
| 备注 |
Brompheniramine hydrogen maleate is a histamine H1 receptors antagonist. |
| 生化机理 |
Brompheniramine Maleate is a histamine H1 receptors antagonist. Brompheniramine Maleate also functions as a moderately effective anticholinergic agent, and is likely an antimuscarinic agent similar to other common antihistamines such as diphenhydramine. Brompheniramine Maleate is an antihistamine drug of the propylamine (alkylamine) class. Brompheniramine Maleate has antidepressant properties, inhibiting reuptake of the neurotransmitter serotonin. Brompheniramine Maleate also has analgesic-sparing (potentiating) effects on opioid analgesics, commonly reducing codeine, dihydrocodeine, and hydrocodone requirements by 10 to 35 percent. Brompheniramine Maleate is metabolised by cytochrome P450s. |
| 别名 |
马来酸溴苯那敏; N,N-二甲基-gamma-(4-溴苯基)-2-吡啶丙胺顺丁烯二酸盐;Bromfed;Brompheniramine maleate; Dimetane maleate;(±)-Brompheniramine maleate salt;1-p-Bromophenyl-1-(2-pyridyl)-3-dimethylaminopropane maleate; 1-(N,N-Dimethylamino)-3-(p-bromophenyl)-3-(alpha-pyridyl)propane maleate |
