货号 | CAS号 |
---|---|
L129692-10mg | 192927-92-7 |
L129692-50mg | 192927-92-7 |
溶解性 |
|
存贮条件 | 储存温度-20°C |
应用 | A selective and potent SR-1D antagonist |
产品介绍 | LY310762是一种5-HT1D受体拮抗剂,Ki为249 nM,对5-HT1B受体具有较低的亲和力。 |
备注 | LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM, having a weaker affinity for 5-HT1B receptor. |
生化机理 | LY-310,762 hydrochloride is a selective and potent SR-1D antagonist. |
别名 | LY 310762; LY-310762; 1-[2-[4-(4-氟苯甲酰基)-1-哌啶基]乙基]-1,3-二氢-3,3-二甲基-2H-吲哚-2-酮盐酸盐;LY-310,762 hydrochloride;LY-310762;1-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-1,3-dihydro-3,3-dimethyl-2H-indol-2-one hydrochloride |