| 应用 |
A compound shown to increase effectiveness of diphenylhydantoin |
| 生化机理 |
Carbetapentane citrate is the citrate form of Carbetapentane. Carbetapentane binds with high affinity to its site in the brain. It has shown to increase the effectiveness of diphenylhydantoin (DPH), a prototypic antiepileptic drug. Additionally reported to be a useful agent in studies of epilepsy treatments. Carbetapentane citrate is an inhibitor of KOR-3 and an activator of σ Receptor 1. |
| 别名 |
托可拉斯; 妥克拉司; 枸橼酸喷托维林;Carbetapentane citrate; 1-Phenylcyclopentanecarboxylic acid 2-(2-diethylaminoethoxy)ethyl ester citrate salt;Carbetapentane citrate salt |
