H 89 2HCl

属性

溶解性	DMSO 104 mg/mL Water 6 mg/mL Ethanol <1 mg/mL
存贮条件	储存温度2-8℃

描述

产品介绍	H 89 2HCl是一种有效的PKA抑制剂，Ki为48 nM，作用于PKA比作用于PKG选择性高10倍，比作用于PKC， MLCK，钙调蛋白激酶II和酪蛋白激I/II选择性高500倍。
备注	H 89 2HCl is a potent PKA inhibitor with Ki of 48 nM, 10-fold selective for PKA than PKG, greater than 500-fold selectivity than PKC, MLCK, calmodulin kinase II and casein kinase I/II.
别名	N-[2-[[3-(4-溴苯基)-2-丙烯-1-基]氨基]乙基]-5-异喹啉磺酰胺盐酸盐(1:2);Protein kinase inhibitor H-89 dihydrochloride; H89 dihydrochloride; H 89 dihydrochloride；N-[2-[[3-(4-Bromophenyl)-2-Propen-1-Yl]Amino]Ethyl]-5-Isoquinolinesulfonamide Hydrochloride (1:2);H-89 Dihydrochloride Hydrate,N-[2-(P-Bromocinnamylamino)Ethyl]-5-Isoquinolinesulfonamide Dihydrochloride; 5-Isoquinolinesulfonamide, N-[2-[[3-(4-Bromophenyl)-2-Propenyl]Amino]Ethyl]-, Dihydrochloride; N-[2-[[3-(4-Bromophenyl)-2-Propen-1-Yl]Amino]Ethyl]-5-Isoquinolinesulfonamide Hydrochloride