应用 |
A potent, non-selective inhibitor of HIV-1 reverse transcriptase. |
产品介绍 |
Nevirapine 是一种非核苷逆转录酶抑制剂(NNRTI),用于治疗HIV-1感染和AIDS。 |
备注 |
Nevirapine(Viramune) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) used to treat HIV-1 infection and AIDS. |
生化机理 |
Nevirapine is a potent (IC50 = 84nM) and selective non-nucleoside inhibitor of HIV-1 reverse transcriptase (HIV-1 RT). |
别名 |
奈韦拉平; 11-环丙基-5,11-二羟基-4-甲基-6H-二吡啶并[3,2-b:2',3'-e][1,4]二氮杂唑-6-酮
;Viramune; BI-RG 587; NSC 641530; NVP;11-Cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-one |