溶解性 | DMSO |
存贮条件 | 储存温度-20°C |
产品介绍 | TAK-715 |
生化机理 |
TAK-715 is a inhibitor of p38 MAPK (IC50 = 7.1 nM for p38 MAPKα). TAK-715 also inhibits Wnt-3a-stimulated β-catenin signaling. Inhibits 22 kinases by more than 80%, including CKIδ/ε. Anti-inflammatory and anti-rheumatoid arthritis agent. Orally bioavailable. |