产品描述
| 溶解性 | DMSO >10 mg/mL |
| 存贮条件 | 储存温度-20°C |
| 生化机理 |
LY2183240 is a novel and highly potent blocker of anandamide uptake (IC50 = 270 pM). LY2183240 inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). Following i.p. administration in rats, LY2183240 increases brain anandamide concentration and exerts antinociceptive effects in formalin model of pain. |
| 别名 | ; |
