产品描述
| 溶解性 | Soluble in water (0.012 mg/ml), DMSO (≥20 mg/ml), methanol, and ethanol (6 mg/ml) |
| 存贮条件 | 储存温度 2-8°C |
| 应用 | A muscarinic receptor antagonist. |
| 产品介绍 | Tolterodine tartrate是Tolterodine的酒石酸盐形式，是一种竞争性的毒蕈碱型乙酰胆碱受体拮抗剂。 |
| 备注 | Tolterodine tartrate (Detrol LA) is a tartrate salt of tolterodine that is a competitive muscarinic receptor antagonist. |
| 生化机理 | Tolterodine L-Tartrate is a muscarinic receptor antagonist that is active at all mAChR M subtypes. This compound blocks the opening of ion channels by acetylcholine, which in turn leads to muscle relaxation by blocking neuronal signaling. Tolterodine L-Tartrate is an inhibitor of mAChR M1, mAChR M2, mAChR M3, mAChR M4 and mAChR M5. |
| 别名 | 酒石酸托特罗定;2-[(1R)-3-[Bis(1-methylethyl)amino]-1-phenylpropyl]-4-methyl-phenol tartrate ;Detrusitol ;PNU-200583E;Detrol LA; Kabi-2234;Tolterodine tartrate |
