溶解性 | DMSO 100 mg/mL Ethanol 100 mg/mL |
存贮条件 | 储存温度-20°C |
产品介绍 | Tofacitinib(CP-690550)是高效JAK3抑制剂,IC50为1 nM,比对JAK2和JAK1的抑制性高20倍和100倍。 |
生化机理 |
Tasocitinib also known as CP690550 is an JAK kinase inhibitor. An IC50 estimated at 0.2 μM for PV patient progenitor cells. |
别名 | (3R,4S)-4-甲基-3-(甲基-7H-吡咯并(2,3-d)嘧啶-4-氨基)-beta-氧代-1-哌啶丙腈; (3R,4S)-托法替尼;(3r,4s)-4-methyl-3-(methyl-7h-pyrrolo(2,3-d)pyrimidin-4-ylamino)-beta-oxo-1-piperidinepropanenitrile |