溶解性 | DMSO 74 mg/mL Water <1 mg/mL Ethanol <1 mg/mL |
存贮条件 | 储存温度-20°C |
产品介绍 | PD168393是一种不可逆的EGFR抑制剂,IC50为0.70 nM,不可逆烷基化Cys-773;抑制insulin, PDGFR, FGFR和PKC活性。 |
备注 | PD168393 is an irreveasible EGFR inhibitor with IC50 of 0.70 nM, irreversibly alkylate Cys-773; inactive against insulin, PDGFR, FGFR and PKC. |
别名 | N-[4-[(3-溴苯基)氨基]-6-喹唑啉基]-2-丙烯酰胺;N-[4-[(3-Bromophenyl)amino]-6-quinazolinyl]-2-propenamide |