产品描述
| 熔点 | 166°C |
| 应用 |
Gabapentin has been used: · as the α2δ-ligand to examine whether the allyl isothiocyanate (AITC) sensitized thermal aversion assay might be useful as a screening method for the identification of presumptive analgesics · dissolved in uptake buffer which is used to measure the to measure ASP (trans-4-[4-(Dimethylamino)styryl]-1-methylpyridinium iodide) substrate by organic cation transporter type 2 (OCTN2) using liquid chromatography - mass spectrometry · used as an analgesic adjuvant for intraperitoneal injections |
| 生化机理 | 具镇惊作用，机制不明;可穿过血脑屏障，增加大脑中的GABA浓度，减少兴奋性氨基酸神经递质，也许是通过其对电压门控钙通道，具有镇痛，抗焦虑药，神经保护，抗痫作用。 |
| 别名 | 加巴喷丁; 1-(氨甲基)环己烷乙酸;1-(甲氨基)环己烷乙酸;Gabapentin; 1-(Aminomethyl)cyclohexaneacetic Acid |
