药物转运蛋白PCR芯片可用于研究表达转运蛋白的84个关键基因的表达。转运蛋白在药理学上发挥了关键作用，影响药物进出细胞进入和排出。对吸收、分布、代谢和排泄重要的转运蛋白包含于芯片。此外，有助于敏感性和抗肿瘤细胞的转运蛋白也在此芯片上。通过实时定量PCR的方法，研究者即能够利用该芯片简单可靠地同时检测与药物转运有关的基因表达。
ABC Transporters: ABCA1, ABCA2, ABCA3, ABCA4, ABCA5, ABCA9, ABCA12, ABCA13, ABCB1 (MDR1), ABCB4, ABCB5, ABCB6, ABCB11, ABCC1 (MRP1), ABCC2 (MRP1), ABCC3 (MRP3), ABCC4, ABCC5 (MRP5), ABCC10, ABCC11, ABCC12, ABCD1, ABCD3, ABCD4, ABCF1, ABCG2 (BCRP), ABCG8, TAP1 (ABCB2), TAP2 (ABCB3). SLC Transporters: SLC2A1, SLC2A2, SLC2A3, SLC3A1, SLC3A2, SLC10A1, SLC10A2, SLC15A1, SLC15A2, SLC16A1, SLC16A2, SLC16A3, SLC19A1, SLC19A2, SLC19A3, SLC22A1, SLC22A2, SLC22A3, SLC22A6, SLC22A7, SLC22A8, SLC22A9, SLC25A13, SLC28A1, SLC28A2, SLC28A3, SLC29A1, SLC29A2, SLC31A1, SLC38A2, SLC38A5, SLC5A1, SLC5A4, SLC7A5, SLC7A6, SLC7A7, SLC7A8, SLC7A9, SLC7A11, SLCO1A2, SLCO1B1, SLCO1B3, SLCO2A1, SLCO2B1, SLCO3A1, SLCO4A1. Other Transporters: Vacuolar H+-ATPase: ATP6V0C. Copper Pumps: ATP7A, ATP7B. Aquaporins: AQP1, AQP7, AQP9. Major Vault Protein: MVP (LRP). Voltage-dependent Anion Channels: VDAC1, VDAC2.