应用 |
A selective SR-4 activator and a SR-3 inhibitor. |
产品介绍 |
Mosapride Citrate是一种促胃肠动力药,是选择性5HT4激动剂。 |
备注 |
Mosapride Citrate is a gastroprokinetic agent that acts as a selective 5HT4 agonist. |
生化机理 |
Mosapride citrate is a selective SR-4 agonist and SR-3 antagonist. Increases gastric emptying in rats and stimulates gastric motor activity in conscious dogs. |
别名 |
枸橼酸莫沙必利; 4-氨基-5-氯-2-乙氧基-N-[[4-(4-氟苄基)-2-吗啉基]甲基]苯甲酰胺枸橼酸盐;Moza citrate; TAK-370 citrate; AS-4370 citrate; Gasmotin citrate;4-Amino-5-chloro-2-ethoxy-N-[[4-[(4-fluorophenyl)methyl]-2-morpholinyl]methyl]-benzamide 2-hydroxy-1,2,3-propanetricarboxylate |