溶解性 | DMSO |
存贮条件 | 储存温度-20°C |
生化机理 |
LY341495(LY 341495; LY-341495) is Highly potent and selective group II metabotropic glutamate receptor antagonist. (Ki/IC50 values are 2.3, 1.3, 173, 990, 6800, 8200 and 22000 nM for human mGlu2, mGlu3, mGlu8 , mGlu7a, mGlu1a, mGlu5a and mGlu4a receptors respectively).LY341495(LY 341495; LY-341495) has readily brain penetrant and active in vivo. |
别名 | ; |